Background
Type: Article

Regioselective synthesis of novel ketene dithioacetals

Journal: Journal of Sulfur Chemistry (17415993)Year: 4 July 2014Volume: 35Issue: Pages: 362 - 372
Habibi A. Valizadeh Y. Alizadeh A.Amiri Rudbari H.a Nardo V.M.
DOI:10.1080/17415993.2013.879871Language: English

Abstract

A series of novel ketene dithioacetals has been synthesized by condensation of active methylene compounds with carbon disulfide in the presence of dialkyl acetylenedicarboxylates. This regioselective reaction provides products in good yield by a Michael addition reaction followed by 5-endo-trig intramolecular cyclization. Structures of synthesized compounds have been characterized by elemental analysis, FT-IR, 1H NMR, 13C NMR, and mass spectra. The crystal structure of compound (C 17H 22O 6S 2) has been determined. © 2014 Taylor & Francis.


Author Keywords

5-endo-trig cyclizationactive methylene compoundsdialkyl acetylenedicarboxylateketene dithioacetalMichael addition

Other Keywords

Addition reactionsCrystal structureCyclizationMass spectrometryRegioselectivity5-endo-trig cyclizationActive methylene compoundsCyclizationsDialkyl acetylenedicarboxylatesDithioacetalsKetene dithioacetalMichael additionsRegioselective reactionsRegioselective synthesisSynthesisedCarbon disulfide